BDBM23408 2-(3,4-dihydroxyphenyl)-3,5,6,7-tetrahydroxy-4H-chromen-4-one::CHEMBL413552::Quercetagetin::Quercetagetin (24)::US11759530, Compound Table1.8
SMILES Oc1ccc(cc1O)-c1oc2cc(O)c(O)c(O)c2c(=O)c1O
InChI Key InChIKey=ZVOLCUVKHLEPEV-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 5 hits for monomerid = 23408
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Loma Linda University School Of Medicine
Curated by ChEMBL
Loma Linda University School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 339nMAssay Description:Inhibition of PIM1 kinaseChecked by AuthorMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Loma Linda University School Of Medicine
Curated by ChEMBL
Loma Linda University School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 340nMAssay Description:Inhibition of Pim1 (unknown origin) assessed as [32P] incorporation preincubated for 15 mins before ATP substrate addition by coupled spectrophotomet...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Loma Linda University School Of Medicine
Curated by ChEMBL
Loma Linda University School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 340nMAssay Description:Inhibition of recombinant PIM1 (unknown origin) expressed in Escherichia coli after 60 mins by ELISAMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Loma Linda University School Of Medicine
Curated by ChEMBL
Loma Linda University School Of Medicine
Curated by ChEMBL
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Loma Linda University School Of Medicine
Curated by ChEMBL
Loma Linda University School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 340nMpH: 7.0 T: 2°CAssay Description:The 96-well flat-bottomed plates were coated with recombinant GST-BAD. After the plates were blocked, the reaction buffer containing test compound an...More data for this Ligand-Target Pair